Pulse Brain · Growing Health Evidence Index
Peer-reviewed

A comprehensive review on the potential of coumarin and related derivatives as multi-target therapeutic agents in the management of gynecological cancers

Gökçe Şeker Karatoprak, Berrak Altınsoy, Engın Celep, İnci Kurt‐Celep, Esra Küpeli Akkol, Eduardo Sobarzo‐Sánchez

Frontiers in Pharmacology · 2024

Read source ↗ All evidence

Summary

Current treatments for gynecological cancers include surgery, radiotherapy, and chemotherapy. However, these treatments often have significant side effects. Phytochemicals, natural compounds derived from plants, offer promising anticancer properties. Coumarins, a class of benzopyrone compounds found in various plants like tonka beans, exhibit notable antitumor effects. These compounds induce cell apoptosis, target PI3K/Akt/mTOR signaling pathways, inhibit carbonic anhydrase, and disrupt microtubules. Additionally, they inhibit tumor multidrug resistance and angiogenesis and regulate reactive oxygen species. Specific coumarin derivatives, such as auraptene, praeruptorin, osthole, and scopoletin, show anti-invasive, anti-migratory, and antiproliferative activities by arresting the cell cycle

Source type
Peer-reviewed study
DOI
10.3389/fphar.2024.1423480
Catalogue ID
SNmoht1vsb-fro4lo
Pulse AI · ask about this record

Dig deeper with Pulse AI.

Pulse AI has read the whole catalogue. Ask about this record, its theme, or how the findings apply to UK farming and policy — every answer cites the underlying studies.