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Peer-reviewed

Targeting Rac and Cdc42 GEFs in Metastatic Cancer

María del Mar Maldonado, Julia I. Medina, Luis Velázquez, Suranganie Dharmawardhane

Frontiers in Cell and Developmental Biology · 2020

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Summary

The Rho family GTPases Rho, Rac, and Cdc42 have emerged as key players in cancer metastasis, due to their essential roles in regulating cell division and actin cytoskeletal rearrangements; and thus, cell growth, migration/invasion, polarity, and adhesion. This review will focus on the close homologs Rac and Cdc42, which have been established as drivers of metastasis and therapy resistance in multiple cancer types. Rac and Cdc42 are often dysregulated in cancer due to hyperactivation by guanine nucleotide exchange factors (GEFs), belonging to both the diffuse B-cell lymphoma (Dbl) and dedicator of cytokinesis (DOCK) families. Rac/Cdc42 GEFs are activated by a myriad of oncogenic cell surface receptors, such as growth factor receptors, G-protein coupled receptors, cytokine receptors, and int

Source type
Peer-reviewed study
DOI
10.3389/fcell.2020.00201
Catalogue ID
SNmoic21xr-5oue13
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