Pulse Brain · Growing Health Evidence Index
Peer-reviewed

Membrane Melatonin Receptors Activated Cell Signaling in Physiology and Disease

Georgi Nikolaev, Ralitsa Robeva, Rossitza Konakchieva

International Journal of Molecular Sciences · 2021

Read source ↗ All evidence

Summary

The pineal hormone melatonin has attracted great scientific interest since its discovery in 1958. Despite the enormous number of basic and clinical studies the exact role of melatonin in respect to human physiology remains elusive. In humans, two high-affinity receptors for melatonin, MT1 and MT2, belonging to the family of G protein-coupled receptors (GPCRs) have been cloned and identified. The two receptor types activate Gi proteins and MT2 couples additionally to Gq proteins to modulate intracellular events. The individual effects of MT1 and MT2 receptor activation in a variety of cells are complemented by their ability to form homo- and heterodimers, the functional relevance of which is yet to be confirmed. Recently, several melatonin receptor genetic polymorphisms were discovered and

Source type
Peer-reviewed study
DOI
10.3390/ijms23010471
Catalogue ID
SNmoj1y55y-fxs0nn
Pulse AI · ask about this record

Dig deeper with Pulse AI.

Pulse AI has read the whole catalogue. Ask about this record, its theme, or how the findings apply to UK farming and policy — every answer cites the underlying studies.