Pulse Brain · Growing Health Evidence Index
Tier 4 — Narrative / commentaryPeer-reviewed

Human Genetics and Genomics for Drug Target Identification and Prioritization: Open Targets’ Perspective

Ellen M. McDonagh, Gosia Trynka, Mark I. McCarthy, Emily Holzinger, Khader Shameer, Nikolina Nakić, Xinli Hu, Helena Cornu, Ian Dunham, David G. Hulcoop

Annual Review of Biomedical Data Science · 2024

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Summary

This paper presents Open Targets' framework for using human genetics and genomics to generate and prioritise therapeutic hypotheses for complex diseases. The consortium integrates large-scale experimental data and informatic platforms to systematically associate genetic variants with drug targets through a multi-evidence approach combining GWAS, functional genomics, epigenetics, rare disease genetics, and experimental perturbation data. The perspective articulates how genetic evidence, when combined with tractability and safety assessments, can accelerate target identification for drug development.

UK applicability

The Open Targets platform incorporates UK Biobank data and is openly accessible to UK-based researchers and industry partners. The methods and predictions may inform UK pharmaceutical research priorities and NHS treatment development strategies, though the framework is international in scope and application.

Key measures

Target prioritisation attributes including clinical precedence, tractability, and safety; locus-to-gene predictions; genome-wide association signals; variant effect predictions; gene burden analyses

Outcomes reported

The study describes Open Targets' integrated informatic platform and methods for systematically building target–disease associations using human genetics and genomic data from multiple large-scale sources including GWAS, UK Biobank, and FinnGen, combined with functional genomic and perturbation data.

Theme
General food systems / other
Subject
Other / interdisciplinary
Study type
Narrative Review
Study design
Narrative review
Source type
Peer-reviewed study
Status
Published
Geography
International
System type
Human clinical
DOI
10.1146/annurev-biodatasci-102523-103838
Catalogue ID
SNmoj1y6jh-6u7muu

Topic tags

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