Pulse Brain · Growing Health Evidence Index
Tier 3 — Observational / field trialPeer-reviewedConventional

Co-formulants in glyphosate-based herbicides disrupt aromatase activity in human cells below toxic levels

Defarge, N., et al

International Journal of Environmental Research and Public Health · 2016

Read source ↗ All evidence

Summary

Pesticide formulations contain declared active ingredients and co-formulants presented as inert and confidential compounds. We tested the endocrine disruption of co-formulants in six glyphosate-based herbicides (GBH), the most used pesticides worldwide. All co-formulants and formulations were comparably cytotoxic well below the agricultural dilution of 1% (18–2000 times for co-formulants, 8–141 times for formulations), and not the declared active ingredient glyphosate (G) alone. The endocrine-disrupting effects of all these compounds were measured on aromatase activity, a key enzyme in the balance of sex hormones, below the toxicity threshold. Aromatase activity was decreased both by the co-formulants alone (polyethoxylated tallow amine—POEA and alkyl polyglucoside—APG) and by the formulations, from concentrations 800 times lower than the agricultural dilutions; while G exerted an effect only at 1/3 of the agricultural dilution. It was demonstrated for the first time that endocrine disruption by GBH could not only be due to the declared active ingredient but also to co-formulants. These results could explain numerous in vivo results with GBHs not seen with G alone; moreover, they challenge the relevance of the acceptable daily intake (ADI) value for GBHs exposures, currently calculated from toxicity tests of the declared active ingredient alone.

Outcomes reported

Pesticide formulations contain declared active ingredients and co-formulants presented as inert and confidential compounds. All co-formulants and formulations were comparably cytotoxic well below the agricultural dilution of 1% (18–2000 times for co-formulants, 8–141 times for formulations), and not the declared active ingredient glyphosate (G) alone. Source report: What Your Food Ate — Montgomery & Biklé (2022), ch.10: SILENT FIELDS Ref#: WYFA-0415 Original: Defarge, N., et al. 2016. Co-formulants in glyphosate-based herbicides disrupt aromatase activity in human cells below toxic levels. International Journal of Environmental Research and Public Health 13:264.

Theme
Farming systems, soils & land use
Subject
Pesticides, contaminants & food safety
Study type
Research
Source type
Peer-reviewed research
Status
Published
Geography
United Kingdom
System type
Other
DOI
10.3390/ijerph13030264
Catalogue ID
IRmqh57rdp-7323e2
Pulse AI · ask about this record

Dig deeper with Pulse AI.

Pulse AI has read the whole catalogue. Ask about this record, its theme, or how the findings apply to UK farming and policy — every answer cites the underlying studies.